DecisionBase PDFs

February 2010

Obesity: A Novel Oral Therapy Emerges That Delivers Superior Weight-Loss Efficacy

Introduction:

Agents entering the obesity market have significant commercial potential thanks to the high prevalence of obesity and the less-than-optimal efficacy and safety of current drugs. Competition in this market will increase significantly over the next ten years as a result of the anticipated launch of several novel therapies for obesity and the loss of patent protection for orlistat (Roche’s Xenical, GlaxoSmithKline’s OTC Alli) and sibutramine (Abbott Laboratories’ Meridia/Reductil). Emerging therapies, in particular  phentermine/topiramate (Vivus’s Qnexa) and Amylin/Takeda’s pramlintide/leptin combination, will come close to satisfying the weight-loss efficacy that physicians and patients expect. Going forward, uptake of these and other novel drugs entering the market will greatly increase the value of the obesity market, which will be approximately seven times greater in 2018 than in 2008. The preliminary findings from the Sibutramine Cardiovascular Outcome Trial (SCOUT), which led to Abbott’s suspension of sibutramine sales in Europe in January 2010, will lead to increased scrutiny of sibutramine in the United States and create more opportunity for emerging agents in European markets.

Questions Answered in This Report:

  *   Weight loss is the most important goal in the treatment of obesity. What are the key primary and secondary clinical trial end points used to evaluate new therapies? How do U.S. and European primary care physicians weight specific efficacy end points and other drug attributes in their prescribing decisions for obesity?

  *   Orlistat is the 2008 major-market sales leader for obesity. How will orlistat and other current therapies fare against emerging therapies? Which drugs do surveyed clinicians anticipate will supplant current therapies? Which agents will suffer the most from competition from emerging agents?

  *   In 2013, phentermine/topiramate (Vivus’s Qnexa) will emerge as the gold-standard therapy in our Drug Comparator Model because of its superior clinical profile compared with the current therapies evaluated in this study. On what clinical attributes is phentermine/topiramate most differentiated from its competitors? Which current therapies are at greatest risk of being replaced by phentermine/topiramate?

Scope:

Key drug development opportunity tested in our target product profiles for obesity: A weight-loss agent that offers greater reduction of fasting blood glucose than orlistat for the treatment of obesity.

Physicians surveyed for this study: 60 U.S. and 31 European primary care physicians.

Comprehensive List of Therapies Included in Our Research and Modeling

Current Therapies

- Orlistat (Roche’s Xenical, GlaxoSmithKline’s OTC Alli)

- Sibutramine (Abbott Laboratories’ Meridia/Reductil)

- Phentermine (GlaxoSmithKline’s Fastin, UCB’s Ionamin, generics)

Emerging Therapies

- Phentermine/topiramate (Vivus’s Qnexa)

- Naltrexone SR/bupropion SR (Orexigen Therapeutics’ Contrave)

- Lorcaserin (Arena Pharmaceuticals)

- Liraglutide (Novo Nordisk’s Victoza)

- Pramlintide/leptin (Amylin Pharmaceuticals/Takeda)

Search Reports

Mentioned in this report:

  • Companies:
  • - Alizyme
  • - Abbott Laboratories
  • - Amylin Pharmaceuticals
  • - Arena Pharmaceuticals
  • - Eisai
  • - Eli Lilly
  • - GlaxoSmithKline
  • - Merck
  • - NeuroSearch
  • - Novartis
  • - Novo Nordisk
  • - Orexigen Therapeutics
  • - Pfizer
  • - Roche
  • - Sanofi-Aventis
  • - Servier
  • - Shionogi
  • - Takeda
  • - Temmler
  • - UCB
  • - Vivus
  • - Wyeth