DecisionBase PDFs

February 2010

Hepatitis C Virus (Treatment Nonresponders): Hope on the Horizon with the Imminent Introduction of HCV-Targeted Therapeutics

Introduction:

Hepatitis C virus (HCV) is an attractive target for drug developers: more than 25 drug candidates are in Phase II development or beyond, representing 9 drug classes. Most of these classes represent novel mechanisms of action for targeting HCV. About half of HCV-infected patients fail treatment, and these HCV treatment nonresponders have few options for subsequent treatment. Thus, an ever-growing portion of HCV-infected patients are sidelined from treatment and await novel therapies that can effectively treat them. Moreover, because the only option for second-line therapy is another round of treatment (with the same therapies that failed the first time) and because of the low relative risk of death associated with HCV, the HCV treatment nonresponder patient population has steadily grown larger over time. Thus, tremendous market potential awaits drugs that can demonstrate improved efficacy in the treatment of this HCV patient subpopulation.

Questions Answered in This Report:

  *   A drug’s performance on at least two efficacy end points, including sustained virologic response, in HCV treatment nonresponders is important for regulatory approval and uptake. What are the key primary and secondary clinical trial end points with which new therapies are evaluated by both regulatory agencies and prescribing clinicians? How do U.S. and European gastroenterologists weight efficacy measures and other drug attributes in their prescribing decisions for treatment of HCV nonresponders?

  *   Peg-IFN-α-2a (Roche’s Pegasys) plus ribavirin (Merck’s Rebetol, Roche’s Copegus, generics) is the 2008 major-market sales leader for the treatment of HCV nonresponders. How will emerging therapies fare against peg-IFN-α-2a/ribavirin? Will emerging therapies offer improvements in the efficacy end points and drug attributes that are most influential in physician prescribing decisions? Which emerging therapies are best positioned to challenge the market-leading status of peg-IFN-α-2a/ribavirin?

  *   In 2013, Vertex/Tibotec/Mitsubishi Tanabe Pharma’s telaprevir (in combination with peg-IFN-α-2a/ribavirin) will emerge as the gold-standard therapy in our Drug Comparator Model because of its superior clinical profile over the current therapies evaluated in this study. On what clinical attributes is telaprevir most differentiated from its competitors?

Scope:

Key drug development opportunity tested in our target product profiles for HCV treatment nonresponders: an HCV-specific antiviral that, when used in combination with peg-IFN-α-2a/ribavirin/telaprevir for 24 weeks, achieves a better SVR than a peg-IFN-α-2a/ribavirin/telaprevir regimen alone for the treatment of nonresponders infected with HCV genotype 1.

Physicians surveyed for this study: 60 U.S. and 32 European gastroenterologists.

Comprehensive List of Therapies Included in Our Research and Modeling

Current Therapies

- Pegylated IFN-α-2a (Roche’s Pegasys)

- Pegylated IFN-α-2b (Merck’s PegIntron)

- IFN-α-con-1 (Three Rivers Pharmaceuticals’ Infergen, Astellas Pharma’s Advaferon)

- Ribavirin (Merck’s Rebetol, Roche’s Copegus, generics)

Emerging Therapies

- Alb-IFN-α-2b (Novartis/Human Genome Sciences’ Zalbin/Joulferon)

- Telaprevir (Vertex/Johnson & Johnson/Misubishi Tanabe Pharma)

- Boceprevir (Merck)

- R-7128 (Roche/Pharmasset)

- TMC-435 (Tibotec)

Search Reports

Mentioned in this report:

  • Companies:
  • - Astellas Pharma
  • - Human Genome Sciences
  • - Intarcia
  • - InterMune
  • - Johnson & Johnson
  • - Merck
  • - Mitsubishi Tanabe Pharma
  • - Nautilus Biotech
  • - Novartis
  • - Pharmasset
  • - Roche
  • - Three Rivers Pharmaceuticals
  • - Tibotec
  • - Valeant
  • - Vertex