Pharmacor

June 2009

Gram-Negative Infections

Report Authors
Hemali Patel, Ph.D.
Jacqueline Lyons, M.P.H.
Alexandra Makarova, M.D., Ph.D.
Danielle L. Drayton, Ph.D.
  • Pages:257
  • Tables:43
  • Figures:11
  • Citations:279
  • Drugs:71
  • Interviews:22

Introduction:

Gram-negative bacteria cause a wide range of infections in both the hospital and community settings. However, because of their pathogenicity and resistance to antibiotics, gram-negative infections (GNIs) acquired in the hospital setting are the most challenging to treat (and are the focus of this report). Hospital-acquired gram-negative infections (GNIs) represent an area of high unmet need and untapped drug development opportunity in the antibacterial market. This market is characterized by rising antibiotic resistance in key gram-negative pathogens (Pseudomonas aeruginosa, Acinetobacter baumannii, Escherichia coli, and Klebsiella pneumoniae), a lean late-stage pipeline, and limited current treatment options. The greatest near-term opportunity in the hospital-acquired GNI market is in the development of agents that can rescue the activity of older antibiotics by countering specific mechanisms of resistance (e.g., beta-lactamase inhibitors). Long-term opportunity lies in the development of a potent antibiotic with a novel mechanism of action that is active against multidrug-resistant gram-negative pathogens.

Questions Answered in This Report:

  *   As many as eight new antibiotics from several existing classes, including cephalosporins, beta-lactam/beta-lactamase inhibitors, carbapenems, and quinolones, have the potential to launch in the next ten years in the hospital-acquired GNI market. What are physicians’ opinions about the clinical potential of these agents? Which emerging agents are most promising? How will these agents be incorporated into medical practice to specifically treat hospital-acquired GNIs? Which of these therapies will have the greatest impact on the hospital-acquired GNI market?

  *   Drug-resistant gram-negative pathogens, such as carbapenemase-producing K. pneumoniae, multidrug-resistant (MDR) Pseudomonas species, and MDR Acinetobacter species are becoming more prevalent and increasingly challenging to treat with the current arsenal of antibiotics. How is medical practice changing for the treatment of such challenging hospital-acquired GNIs? How will emerging therapies address these challenges? What prescribing trends do physicians expect to see in the coming years?

  *   A few highly potent, broad-spectrum branded antibiotics—Wyeth’s Zosyn/Tazocin, Johnson & Johnson’s Levaquin, Merck’s Primaxin, and Cubist Pharmaceuticals/AstraZeneca’s Merrem/Meronem—have fueled growth in the GNI market over the past ten years. Expected patent expiries of these products may allow entry of generics during the 2008-2018 forecast period. To what extent will generic erosion of these key products affect sales in the hospital-acquired GNI market? Will emerging therapies be able to recoup lost sales of leading brands? Which classes will continue to be commercially successful in the face of generic competition?

  *   The pipeline of therapies in early-stage development comprises a variety of interesting new classes and novel approaches for the treatment of hospital-acquired GNIs, including antibodies against drug-resistant, nosocomial gram-negative pathogens (e.g., P. aeruginosa). How receptive are physicians to such approaches? What are the most promising early-stage therapies in the pipeline for hospital-acquired GNIs?

Scope:

Markets covered: United States, France, Germany, Italy, Spain, United Kingdom, Japan.

Primary research: 22 country-specific interviews with thought leaders.

Epidemiology: Diagnosed events of hospital-acquired infections in the major pharmaceutical markets; estimates of gram-negative drug-treated populations in the major pharmaceutical markets.

Population segments in market forecast: Urinary tract infections, nosocomial pneumonia (includes hospital-acquired and healthcare-associated pneumonia), bloodstream infections, complicated skin and skin structure infections/surgical site infections.

Emerging therapies: Phase II: 10 drugs; Phase III: 3 drugs; preregistration: 1 drug; registered: 2 drugs. Coverage of 31 select preclinical and Phase I products.

Market forecast features: Using data from the Arlington Medical Resources, Inc. (AMR; a Decision Resources company), Hospital Antibiotic Market Guide, we estimate the number of patients currently treated in a hospital setting with an antibiotic that is active against gram-negative pathogens. This approach informs our estimates for size of the candidate population that can be targeted by current and emerging agents in the GNI market.

Search Reports

Mentioned in this report:

  • Abbott Laboratories
  • Achaogen
  • Alliance Pharmaceutical Corporation
  • Aridis
  • Arpida
  • Astellas Pharma
  • AstraZeneca
  • AvidBiotics
  • Basilea Pharmaceutica
  • Bayer Healthcare
  • Bioline Innovations
  • Bristol-Myers Squibb
  • Cadence Pharmaceuticals
  • Calixa
  • Ceragenix Pharmaceuticals
  • Cerexa
  • Chiron
  • Combinature Biopharm
  • ConjuGon
  • Cubist Pharmaceuticals
  • Daiichi Sankyo
  • Dainippon Sumitomo Pharma
  • Demegen
  • Dura Pharmaceuticals
  • Elan
  • Eli Lilly
  • Forest Laboratories
  • Gilead Sciences
  • GlaxoSmithKline
  • Immunsystem
  • Intercell
  • Janssen-Cilag
  • Johnson & Johnson
  • KaloBios Pharmaceuticals
  • Kenta Biotech
  • Lek
  • Lytix Biopharma
  • Meiji Seika Kaisha
  • Merck & Co.
  • MerLion Pharmaceuticals
  • Microbiotix
  • Migenix
  • Mpex Pharmaceuticals
  • Nektar Therapeutics
  • Northern Antibiotics
  • NovaBay Pharma
  • Novartis
  • Novexel
  • Novozymes
  • Ortho-McNeil
  • Oscient Pharmaceuticals
  • Paratek Pharmaceuticals
  • Pelias
  • Pfizer
  • PolyMedix
  • Polyphor
  • Procter & Gamble
  • Protez Pharmaceuticals
  • Quotient BioResearch
  • Replidyne
  • Rib-X Pharmaceuticals
  • Roche
  • Sandoz
  • Sanofi-Aventis
  • Schering-Plough
  • Shionogi
  • Spider Biotech
  • TaiGen Biotechnology
  • Takeda Pharmaceutical
  • Targanta
  • The Medicines Company
  • Theravance
  • Transave
  • Wakunaga Pharmaceutical
  • Wockhardt
  • Wyeth